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nmpa_approved_drug_library
/library/nmpa_approved_drug_library
NMPA中国上市药物库
NMPA-Approved Drug Library
产品编号: L4210

NMPA 中国上市药物库汇集了 1319 个中国国家药品监督管理局批准的化合物,所有化合物通过临床验证,靶点明确,具有较好的安全性和生物利用度,是进行老药新用理想的工具,可以大大提高药物研发的成功率,能够缩短药物研发周期,节约研发成本。

陶术生物的所有产品和服务仅用于科学研究,我们不为任何个人用途提供产品和服务。
产品规格
  • 1319个NMPA批准药物的独特集合,可用于高通量筛选和高内涵筛选;
  • 全部得到NMPA批准,提供NMPA批准编号,用于药物重定位、新的药物靶点筛选的有效工具;
  • 经过了严格的临床前研究和临床试验,生物活性和安全性得到保障;
  • 涵盖多个研究领域:肿瘤、心血管药物、抗炎、免疫、神经系统药物、呼吸系统药物等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。
化合物库定制
我们的化合物库可以灵活定制!了解更多
化合物库咨询
化合物库组成
Antibacterial (228)
Antibiotic (225)
Autophagy (197)
Endogenous Metabolite (142)
Apoptosis (132)
Adrenergic Receptor (91)
5-HT Receptor (87)
COX (68)
AChR (66)
Histamine Receptor (55)
DNA/RNA Synthesis (53)
Dopamine Receptor (53)
Calcium Channel (48)
Antifungal (44)
Parasite (43)
Sodium Channel (43)
Potassium Channel (40)
Topoisomerase (40)
HIV Protease (35)
Glucocorticoid Receptor (33)
Ferroptosis (28)
NF-κB (26)
Influenza Virus (25)
Reactive Oxygen Species (25)
Estrogen/progestogen Receptor (24)
RAAS (23)
Nucleoside Antimetabolite/Analog (22)
P450 (22)
PDE (20)
Mitophagy (19)
ribosome (18)
Antifection (17)
EGFR (17)
Serotonin Transporter (17)
GABA Receptor (16)
HSV (16)
Reverse Transcriptase (16)
AChE (15)
Dehydrogenase (15)
Microtubule Associated (15)
PDGFR (15)
PPAR (15)
HBV (14)
Prostaglandin Receptor (14)
SARS-CoV (14)
c-Kit (13)
DNA Alkylator/Crosslinker (13)
Opioid Receptor (13)
iGluR (12)
Proton pump (12)
Virus Protease (12)
ATPase (11)
Norepinephrine (11)
VEGFR (11)
Androgen Receptor (10)
MRP (10)
ROS (10)
TNF (10)
Estrogen Receptor/ERR (9)
IL Receptor (9)
Phospholipase (9)
TRP/TRPV Channel (9)
Antifolate (8)
Bcr-Abl (8)
CaMK (8)
HMG-CoA Reductase (8)
Progesterone Receptor (8)
Proteasome (8)
Adenosine Receptor (7)
Amino Acids and Derivatives (7)
DHFR (7)
FGFR (7)
HIF/HIF Prolyl-Hydroxylase (7)
MAO (7)
Mitochondrial Metabolism (7)
NMDAR (7)
Thyroid hormone receptor(THR) (7)
AMPK (6)
Carbonic Anhydrase (6)
GluR (6)
HCV Protease (6)
Interleukin (6)
NO Synthase (6)
Phosphatase (6)
PKC (6)
Retinoid Receptor (6)
Antioxidant (5)
CAT (5)
c-Met/HGFR (5)
DNA Alkylation (5)
DNA gyrase (5)
MMP (5)
P-gp (5)
STAT (5)
ABC (4)
ALK (4)
Antiviral (4)
Aromatase (4)
Beta Amyloid (4)
FLT (4)
HER (4)
Histone Methyltransferase (4)
Monoamine Oxidase (4)
Raf (4)
Src (4)
Thrombin (4)
Xanthine Oxidase (4)
AhR (3)
Annexin A (3)
Anti-infection (3)
Caspase (3)
CDK (3)
c-RET (3)
DNA Methyltransferase (3)
DPP-4 (3)
Drug Metabolite (3)
ERK (3)
Factor Xa (3)
Fatty Acid Synthase (3)
Free radical scavengers (3)
Glucosidase (3)
Glutathione Peroxidase (3)
GNRH Receptor (3)
GPR (3)
HDAC (3)
HSP (3)
Imidazoline Receptor (3)
Lipoxygenase (3)
LTR (3)
P2Y Receptor (3)
PKA (3)
Reductase (3)
Sigma receptor (3)
TGF-beta/Smad (3)
TLR (3)
Transferase (3)
Vasopressin Receptor (3)
Wnt/beta-catenin (3)
Adenosine deaminase (2)
Akt (2)
Aminopeptidase (2)
BCL (2)
CaSR (2)
CFTR (2)
Chloride channel (2)
Cysteine Protease (2)
DNA (2)
Endothelin Receptor (2)
FXR (2)
GST (2)
HIF (2)
IRE1 (2)
IκB/IKK (2)
Leukotriene Receptor (2)
Ligand for E3 Ligase (2)
MEK (2)
Melatonin Receptor (2)
Molecular Glues (2)
mTOR (2)
NADPH (2)
Neprilysin (2)
NOD (2)
NOD-like Receptor (NLR) (2)
NOS (2)
Oxytocin Receptor (2)
P2X Receptor (2)
p38 MAPK (2)
PARP (2)
PGE Synthase (2)
Rho (2)
ROS Kinase (2)
Serine Protease (2)
TOPK (2)
Trk receptor (2)
Tyrosine Kinases (2)
Acyltransferase (1)
advanced glycation end products (1)
Arginase (1)
Aryl Hydrocarbon Receptor (1)
Aurora Kinase (1)
BACE (1)
BTK (1)
Cannabinoid Receptor (1)
CCR (1)
CGRP Receptor (1)
cholecystokinin (1)
Complement System (1)
CRISPR/Cas9 (1)
Decarboxylase (1)
Ephrin Receptor (1)
Epigenetic Reader Domain (1)
Epoxide Hydrolase (1)
Gap Junction Protein (1)
Glucagon Receptor (1)
Glutathione reductase (1)
GPCR19 (1)
GRK (1)
GSK-3 (1)
Guanylate cyclase (1)
Hedgehog/Smoothened (1)
Histone Demethylase (1)
Hydrogenase (1)
Hydroxylase (1)
Indoleamine 2,3-Dioxygenase (IDO) (1)
Integrase (1)
Integrin (1)
JAK (1)
LDL (1)
Lipase (1)
Lipid (1)
Mdm2 (1)
Monoamine Transporter (1)
Monocarboxylate transporter (1)
MT Receptor (1)
Na+/Ca2+ Exchanger (1)
NADPH-oxidase (1)
Na-K-Cl cotransporter (1)
Neurokinin receptor (1)
Nrf2 (1)
PAFR (1)
PI3K (1)
RAR/RXR  (1)
Ras (1)
ROCK (1)
ROR (1)
RSV (1)
S6 Kinase (1)
Serine/threonin kinase (1)
Sirtuin (1)
Smo (1)
Telomerase (1)
Tyrosinase (1)
化合物库信息示例
Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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