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Glucokinase
T0247 Acarbose Acarbose is an inhibitor of α-Glucosidases with antihyperglycemic activity.
T0714 Oxfendazole Oxfendazole, a broad spectrum benzimidazole anthelmintic,protects livestock against roundworm, strongyles and pinworms.
T2455 PFK-015 PFK-015 is an effective inhibitor of PFKFB3 (IC50: 110 nM) and inhibits PFKFB3 activity in Y cells (IC50: 20 nM).
T3104 LY2608204 LY2608204 has been used in trials studying the treatment of Diabetes Mellitus, Type 2.
T3105 PFK-158 PFK-158 is an effective and specific inhibitor PFKFB3.
T3260 3PO 3PO is a PFKFB3 (6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase) inhibitor.
T3312 AM-2394 AM-2394 is an effective and specific Glucokinase agonist (GKA, EC50: 60 nM), which catalyzes the phosphorylation of glucose to glucose-6-phosphate. AM-2394 increases the affinity of GK for glucose by approximately 10-fold, exhibits moderate clearance and good oral bioavailability in multiple animal
T3386 Kaempferitrin Kaempferitrin has antidepressant-like effect related to the serotonergic system, principally 5-HT1A. Kaempferitrin exerts cytotoxic and antitumor effects against HeLa cells. Kaempferitrin stimulates glucose-metabolizing enzymes, promotes glucose homeostasis. Kaempferitrin exerts immunostimulatory e
T3871 Eleutheroside A Eleutheroside A (Daucosterol) has proliferation-enhancing activity, may be involved in the IGF1-AKT pathway. Daucosterol has efficient and inexpensive neuroprotectant effect, to contribute to IGF1-like activity, could be potentially developed as a medicine for ischemic stroke treatment.
T4049 Genz 123346 Genz 123346 is an inhibitor of GL1 synthase that blocks the conversion of ceramide to GL1.
T6723 Voglibose Voglibose, an N-substituted derivative of valiolamine, exhibits excellent inhibitory activity against α-glucosidases and action against hyperglycemia and various disorders caused by hyperglycemia.
T6759 AP-III-a4 (ENOblock) AP-III-a4 (ENOblock) is the first nonsubstrate analogue inhibitor of enolase with IC50 of 0.576 μM.
T4280 LTI-291 LTI-291 is a glucocerebrosidase (Gcase) activator.
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